European Patent Office

T 0643/96 (Bioisosterism/BEECHAM) of 14.10.1996

European Case Law Identifier
ECLI:EP:BA:1996:T064396.19961014
Date of decision
14 October 1996
Case number
T 0643/96
Petition for review of
-
Application number
88312038.8
IPC class
C07D 453/02
Language of proceedings
English
Distribution
Distributed to board chairmen and members (B)
OJ versions
No OJ links found
Other decisions for this case
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Abstracts for this decision
-
Application title
Azabicyclic compounds, process for their preparation and pharmaceutical compositions containing them
Applicant name
BEECHAM GROUP PLC
Opponent name
-
Board
3.3.01
Headnote
-
Keywords
Inventive step - yes - chemical compounds - no pointer to claimed compounds
Catchword
1. The concept of bioisosterism has to be applied with caution when deciding upon inventive step (No. 4.2.3.3).
2. When deciding upon inventive step in relation to pharmacologically active compounds, what is essential is not whether a particular substructure of a chemical compound is replaced by another known isosteric one, but whether information was available on the impact of such a replacement on the pharmacological activity profile of the specific (group of) compound(s) concerned (No. 4.2.3.5).

ORDER

for these reasons it is decided that:

1. The decision under appeal is set aside.

2. The case is remitted to the Examining Division with the order to grant a patent on the basis of the following documents:

- Claims 1 to 11 for all the designated contracting states except Spain, as filed by fax on 13. September 1996;

- Claims 1 to 8 for Spain, as filed by fax on 13. September 1996;

- a description to be adapted accordingly.